美国药品专利与行政保护速查

Abacavir sulfate(硫酸阿巴卡韦)1

Abacavir sulfate （硫酸阿巴卡韦）;lamivudine（拉米夫定）1

Abacavir sulfate （硫酸阿巴卡韦）;lamivudine（拉米夫定）；zidovudine （齐多夫定）1

Abarelix(阿巴瑞克)2

Abiraterone acetate（醋酸阿比特龙酯）2

Acetaminophen(对乙酰氨基酚)3

Acetaminophen(对乙酰氨基酚)； aspirin（阿司匹林）;caffeine（咖啡因）3

Acetylcholine chloride(氯化乙酰胆碱)3

Acetylcysteine(乙酰半胱氨酸)4

Aclidinium bromide(阿地溴铵)4

Acyclovir（阿昔洛韦）;hydrocortisone(氢化可的松)4

Adapalene(阿达帕林)5

Adapalene(阿达帕林);benzoyl peroxide(过氧化苯甲酰)5

Adefovir dipivoxil(阿德福韦酯)6

Adenosine(腺苷)6

Alatrofloxacin mesylate(甲磺酸阿拉曲伐沙星)6

Albumin Human(人白蛋白)7

Albuterol sulfate(硫酸沙丁胺醇)7

Albuterol sulfate(硫酸沙丁胺醇);ipratropium bromide(溴化异丙托品)8

Alcaftadine(阿卡他定)9

Alcohol(酒精);chlorhexidine gluconate(葡萄糖酸氯己定)9

Alendronate sodium(阿仑膦酸钠)10

Alendronate sodium（阿仑膦酸钠）;cholecalciferol （胆钙化醇）11

Alfuzosin hydrochloride(盐酸阿夫唑嗪)11

Aliskiren Hemifumarate(阿利克仑半富马酸盐)12

Aliskiren hemifumarate （阿利克仑半富马酸）;amlodipine besylate （苯磺酸氨氯地平）12

Aliskiren hemifumarate （阿利克仑半富马酸）;amlodipine besylate （苯磺酸氨氯地平）;hydrochlorothiazide（氢氯噻嗪）13

Aliskiren hemifumarate （阿利克仑半富马酸）;hydrochlorothiazide（氢氯噻嗪）13

Aliskiren hemifumarate （阿利克仑半富马酸）;valsartan （缬沙坦）14

Alitretinoin （阿利维甲酸）14

Almotriptan malate(苹果酸阿莫曲普坦)15

Alosetron hydrochloride(盐酸阿洛司琼)15

Alprazolam(阿普唑仑)15

Alprostadil(前列地尔)16

Alvimopan(爱维莫潘)16

Ambrisentan（安贝生坦）17

Amifostine(氨磷汀)17

Aminolevulinic acid hydrochloride(盐酸氨基酮戊酸)18

Amiodarone hydrochloride(盐酸胺碘酮)18

Amlodipine besylate(苯磺酸氨氯地平)18

Amlodipine besylate（苯磺酸氨氯地平）;atorvastatin calcium(阿托伐他汀钙)19

Amlodipine besylate （苯磺酸氨氯地平）;hydrochlorothiazide（氢氯噻嗪）;olmesartan medoxomil(奥美

沙坦酯)21

Amlodipine besylate （苯磺酸氨氯地平）;hydrochlorothiazide（氢氯噻嗪）;valsartan(缬沙坦)21

Amlodipine besylate （苯磺酸氨氯地平）;olmesartan medoxomil(奥美沙坦酯)22

Amlodipine besylate （苯磺酸氨氯地平）;telmisartan(替米沙坦)23

Amlodipine besylate （苯磺酸氨氯地平）;valsartan(缬沙坦)23

Amoxicillin(阿莫西林)24

Amoxicillin（阿莫西林）;clavulanate potassium(克拉维酸钾)24

Amphetamine aspartate （天门冬氨酸苯丙胺）;amphetamine sulfate （硫酸苯丙胺）;dextroamphetamine

saccharate（糖酸右苯丙胺）;dextroamphetamine sulfate（硫酸右苯丙胺）24

Amphotericin B(两性霉素B)27

Amprenavir(安普那韦)27

Anidulafungin(阿尼芬净)28

Apixaban(阿哌沙班)28

Aprepitant(阿瑞吡坦)28

Arformoterol tartrate(酒石酸阿福莫特罗)29

Argatroban(阿加曲班)29

Aripiprazole(阿立哌唑)30

Armodafinil(阿莫达非尼)31

Arsenic trioxide(三氧化砷)32

Artemether（蒿甲醚）;lumefantrine(苯芴醇)32

Ascorbic acid （抗坏血酸）;polyethylene glycol 3350 （聚乙二醇3350）;potassium chloride;sodium

ascorbate （抗坏血酸钠）;sodium chloride（氯化钠）;sodium sulfate(硫酸钠)33

Asenapine maleate(马来酸阿塞那平)33

Aspirin(阿司匹林),dipyridamole(双嘧达莫)34

Aspirin(阿司匹林);pravastatin sodium(普伐他汀钠)34

Atazanavir sulfate(硫酸阿扎那韦)35

Atomoxetine hydrochloride(盐酸阿托莫西汀)35

Atorvastatin calcium(阿伐他汀钙)36

Atovaquone(阿托伐醌)37

Atovaquone(阿托伐醌);proguanil hydrochloride(盐酸氯胍)37

Avanafil （阿伐那非）38

Axitinib(阿西替尼)38

Azelaic acid(壬二酸)39

Azelastine hydrochloride(盐酸氮卓斯汀)39

Azelastine hydrochloride(盐酸氮卓斯汀);fluticasone propionate(丙酸氟替卡松) 39

Azilsartan kamedoxomil(阿齐沙坦酯)40

Azilsartan kamedoxomil(阿齐沙坦酯);chlorthalidone(氯噻酮)40

Azithromycin(阿奇霉素)41

Aztreonam(氨曲南)42

Baclofen(巴氯芬)42

Balsalazide disodium(巴柳氮二钠)42

Beclomethasone dipropionate(丙酸倍氯米松)43

Bedaquiline fumarate(富马酸巴达喹啉)44

Benzoyl peroxide（过氧化苯甲酰）;clindamycin phosphate（磷酸克林霉素）44

Benzyl alcohol(苯甲醇)44

Bepotastine besilate(苯磺贝他斯汀)45

Besifloxacin hydrochloride(盐酸贝西沙星)45

Betamethasone dipropionate(二丙酸倍他米松);calcipotriene hydrate(卡泊三醇水合物)45

Betamethasone valerate(戊酸倍他米松)46

Betaxolol hydrochloride（盐酸倍他洛尔）;pilocarpine hydrochloride(盐酸毛果芸香碱)46

Bexarotene（蓓萨罗丁）47

Bimatoprost(贝美前列素)47

Bisacodyl （比沙可啶）;polyethylene glycol 3350 （聚乙二醇3350）;potassium chloride（氯化钾）;sodium

bicarbonate（碳酸氢钠）;sodium chloride(氯化钠)48

Bismuth subcitrate potassium（枸橼酸铋钾）;metronidazole（甲硝唑）;tetracycline hydrochloride(盐酸

四环素)48

Bivalirudin(比伐卢定)49

Boceprevir(包西普韦)49

Bortezomib(硼替佐米)50

Bosentan(波生坦)50

Bosutinib monohydrate(博舒替尼)51

Brimonidine tartrate(酒石酸溴莫尼定)51

Brimonidine tartrate（酒石酸溴莫尼定);timolol maleate(马来酸噻吗洛尔)52

Bromocriptine mesylate(甲磺酸溴隐亭)52

Budesonide(布地奈德)53

Budesonide(布地奈德);formoterol fumarate dihydrate(富马酸福莫特罗二水物)54

Bupivacaine（布比卡因）55

Buprenorphine（丁丙诺啡）55

Buprenorphine（丁丙诺啡）;naloxone(纳洛酮)56

Bupropion hydrobromide(氢溴酸安非他酮)56

Busulfan(白消安)58

Butoconazole nitrate(硝酸布康唑)58

Cabazitaxel(卡巴他赛)58

Cabozantinib smalate(苹果酸卡波替尼)59

Calcipotriene(卡泊三烯)59

Calcitonin salmon(鲑鱼降钙素)60

Calcitonin salmon recombinant(鲑鱼降钙素重组蛋白)60

Calcitriol(骨化三醇)61

Calcium acetate（醋酸钙）61

Calcium carbonate(碳酸钙);famotidine(法莫替丁);magnesium hydroxide(氢氧化镁)62

Calcium carbonate（碳酸钙）;risedronate sodium（利塞膦酸钠）62

Calcium chloride （氯化钙）;dextrose（葡萄糖）;magnesium chloride（氯化镁）;oxiglutatione （奥谷胱

甘肽）;potassium chloride （氯化钾）;sodium bicarbonate （碳酸氢钠）;sodium chloride （氯化钠）;

sodium phosphate(磷酸钠)63

Candesartan cilexetil(坎地沙坦酯)63

Candesartan cilexetil(坎地沙坦酯)；hydrochlorothiazide（氢氯噻嗪）64

Capecitabine（卡培他滨）65

Capsaicin（辣椒素）65

Carbamazepine(卡马西平)65

Carbidopa(卡比多巴) ;entacapone(恩他卡朋);levodopa(左旋多巴)66

Carfilzomib (卡菲佐米)67

Carvedilol (卡维地洛)67

Carvedilol phosphate (磷酸卡维地洛)68

Caspofungin acetate(醋酸卡泊芬净)69

Cefditoren pivoxil(头孢妥仑匹酯)69

Ceftaroline fosamil(头孢他洛林酯)70

Ceftibuten dihydrate(头孢布烯二水合物)70

Celecoxib(塞来昔布)70

Cetirizine hydrochloride(盐酸西替利嗪)71

Cetirizine hydrochloride(盐酸西替利嗪)；pseudoephedrine hydrochloride（盐酸右旋麻黄素）72

Cetrorelix（西曲瑞克）72

Chlorhexidine gluconate(葡萄糖酸氯己定)72

Chlorhexidine gluconate （葡萄糖酸氯己定）;isopropyl alcohol(异丙醇)73

Chlorpheniramine maleate(马来酸氯苯那敏),ibuprofen(布洛芬),pseudoephedrine hydrochloride

(盐酸伪麻黄碱)74

Choline fenofibrate(非诺贝特胆碱)75

Choriogonadotropin alfa(重组人绒促性素)75

Ciclesonide(环索奈德)75

Cinacalcet hydrochloride(盐酸西那卡塞)76

Ciprofloxacin(环丙沙星);ciprofloxacin hydrochloride(盐酸环丙沙星)77

Ciprofloxacin(环丙沙星);dexamethasone（地塞米松）78

Cisapride monohydrate（西沙必利水合物）78

Clarithromycin(克拉霉素)79

Clevidipine butyrate(丁酸氯维地平)79

Clindamycin phosphate(克林霉素磷酸酯)79

Clindamycin phosphate(克林霉素磷酸酯)；tretinoin（维甲酸）80

Clobetasol propionate（丙酸氯倍）80

Clofarabine(氯法拉滨)81

Clopidogrel bisulfate(硫酸氢氯吡格雷)81

Clozapine(氯氮平)82

Cobicistat（柯比西替）;elvitegravir（埃维替韦）;emtricitabine（恩曲他滨）;tenofovir disoproxil

fumarate(富马酸替诺福韦)83

Colchicine(秋水仙碱)83

Colesevelam hydrochloride(盐酸考来维仑)84

Conivaptan hydrochloride （盐酸考尼伐坦）86

Crizotinib(克里唑替尼)87

Crofelemer(克罗非马)87

Cyanocobalamin(氰钴胺)87

Cyclobenzaprine hydrochloride(盐酸环苯扎林)88

Cyclosporine(环孢素)88

Dabigatran etexilate mesylate(达比加群酯甲磺酸盐)89

Dalfampridine(氨基吡啶)89

Dapsone (氨苯砜)90

Daptomycin (达托霉素)90

Darifenacin hydrobromide (氢溴酸达非那新)91

Darunavir ethanolate (地瑞那韦乙醇)91

Dasatinib (达沙替尼)96

Deferasirox (地拉罗斯)97

Degarelix acetate (地加瑞克)98

Delavirdine mesylate (甲磺酸地拉韦啶)98

Desflurane (去氟烷)98

Desirudin recombinant (重组地西卢定)99

Desloratadine (地氯雷他定)99

Desloratadine（地氯雷他定）;pseudoephedrine sulfate (硫酸伪麻黄碱)100

Desmopressin acetate (醋酸去氨加压素)101

Desonide (地奈德)102

Desvenlafaxine succinate (琥珀酸去甲文拉法辛)103

Dexamethasone (地塞米松)103

Dexamethasone(地塞米松);tobramycin (妥布霉素)104

Dexlansoprazole (右兰索拉唑)104

Dexmedetomidine hydrochloride (盐酸右美托咪定)106

Dexrazoxane hydrochloride (盐酸右雷佐生)107

Dextromethorphan hydrobromide(氢溴酸右美沙芬);guaifenesin (愈创甘油醚)108

Dextromethorphan hydrobromide (氢溴酸右美沙芬）;quinidine sulfate (硫酸奎尼丁)108

Dextromethorphan polistirex (右美沙芬聚合物)109

Diazepam (地西泮)109

Diclofenac potassium (双氯芬酸钾)109

Diclofenac sodium (双氯芬酸钠)；misoprostol （米索前列醇）110

Dienogest (地诺孕素);estradiol valerate (戊酸雌二醇)111

Difluprednate (二氟泼尼酯)111

Diltiazem hydrochloride (盐酸地尔硫卓)111

Dimyristoyl lecithin（二棕榈酰卵磷酯）;perflexane (全氟己烷)112

Diphenhydramine citrate （枸橼酸苯海拉明）;ibuprofen (布洛芬)113

Divalproex sodium (双丙戊酸钠)113

Docetaxel (多西他赛)114

Docosanol (二十二醇)115

Dofetilide (多非利特)115

Donepezil hydrochloride (盐酸多奈哌齐)115

Doripenem (多尼培南)116

Doxepin hydrochloride (盐酸多塞平)116

Doxercalciferol (度骨化醇)117

Doxycycline (多西环素)117

Doxycycline hyclate (多西环素盐酸乙醇水合物)118

Dronedarone hydrochloride (盐酸决奈达隆)118

Drospirenone(屈螺酮);estradiol (雌二醇)119

Drospirenone(屈螺酮);ethinyl estradiol (乙炔雌二醇)119

Drospirenone（屈螺酮）;ethinyl estradiol（炔雌醇）;levomefolate calcium (左甲基四氢叶酸钙)119

Duloxetine hydrochloride (盐酸度洛西汀)120

Dutasteride（度他雄胺）;tamsulosin hydrochloride (盐酸坦索罗辛)121

Efavirenz (依法韦恩茨)122

Efavirenz(依法韦恩茨);emtricitabine (恩曲他滨);tenofovir disoproxil fumarate (替诺福韦酯富马

酸盐)123

Eflornithine hydrochloride (盐酸依氟鸟氨酸)124

Eletriptan hydrobromide (依来曲普坦氢溴酸盐)124

Eltrombopag olamine (艾曲波帕)125

Emtricitabine（恩曲他滨）127

Emtricitabine（恩曲他滨）;rilpivirine（利匹韦林）;tenofovir disoproxil fumarate (替诺福韦酯富马

酸盐)127

Enfuvirtide(恩夫韦肽)129

Entacapone (恩他卡朋)129

Entecavir (恩替卡韦)129

Enzalutamide ( 恩扎罗酰胺)130

Epinephrine (肾上腺素)130

Epinephrine (肾上腺素)；lidocaine hydrochloride (盐酸利多卡因)131

Eplerenone (依普利酮)131

Epoprostenol sodium (依前列醇钠)133

Eprosartan mesylate (依普罗沙坦甲磺酸盐)134

Eprosartan mesylate（依普罗沙坦甲磺酸盐）;hydrochlorothiazide (氢氯噻嗪)134

Eptifibatide (依非巴特)134

Eribulin mesylate (甲磺酸艾日布林)135

Erlotinib hydrochloride (盐酸厄洛替尼)135

Ertapenem sodium(厄他培南钠)136

Escitalopram oxalate (草酸依地普仑)136

Esmolol hydrochloride (盐酸艾司洛尔)137

Esomeprazole magnesium（埃索美拉唑镁）138

Esomeprazole magnesium（埃索美拉唑镁）;naproxen (萘普生)142

Esomeprazole sodium（埃索美拉唑钠） 143

Estradiol (雌二醇)143

Estradiol acetate (醋酸雌二醇)144

Estradiol hemihydrate ( 雌二醇半水合物)145

Estradiol（雌二醇）;levonorgestrel (左炔诺孕酮)145

Estradiol（雌二醇）;norethindrone acetate (炔诺酮醋酸酯)145

Estradiol（雌二醇）;norgestimate (诺孕酯)146

Estrogens, conjugated synthetic a (组合雌激素a)146

Estrogens, conjugated synthetic b (组合雌激素b) 146

Estrogens, conjugated （组合雌激素）;medroxyprogesterone acetate (醋酸甲羟孕酮)147

Eszopiclone (艾司佐匹克隆)148

Ethinyl estradiol （炔雌醇);etonogestrel(依托孕烯)148

Ethinyl estradiol （炔雌醇）;levonorgestrel (左炔诺孕酮)148

Ethinyl estradiol(炔雌醇);norethindrone (炔诺酮)149

Ethinyl estradiol(炔雌醇);norgestimate (诺孕酯)149

Etravirine (依曲韦林)150

Everolimus (依维莫司)150

Exenatide synthetic (合成艾塞那肽)153

Ezetimibe (依泽替米贝)154

Ezetimibe(依泽替米贝)；simvastatin (辛伐他汀)154

Famciclovir (泛昔洛韦)155

Famotidine (法莫替丁)156

Famotidine(法莫替丁);ibuprofen (布洛芬)157

Febuxostat (非布索坦)157

Fenofibrate (非诺贝特)157

Fenofibric acid (非诺贝酸)158

Fentanyl citrate (枸橼酸芬太尼)159

Fentanyl hydrochloride (盐酸芬太尼 )161

Ferumoxytol (菲立氧铁)161

Fesoterodine fumarate (富马酸非索罗定)161

Fexofenadine hydrochloride (盐酸非索非那定)162

Fexofenadine hydrochloride（盐酸非索非那定）;pseudoephedrine hydrochloride (盐酸伪麻黄碱)165

Fidaxomicin (非达霉素)166

Finasteride (非那雄胺)167

Fingolimod (芬戈莫德)167

Florbetapir F18（氟罗贝它 F18）167

Fludarabine phosphate (磷酸氟达拉滨)168

Flunisolide (氟尼缩松)168

Fluocinolone acetonide (氟新诺龙丙酮)168

Fluocinolone acetonide (氟新诺龙丙酮)；hydroquinone（氢醌）;tretinoin（维甲酸）169

Fluocinonide (醋酸氟轻松)169

Fluorouracil (氟脲嘧啶)169

Fluoxetine hydrochloride（盐酸氟西汀）170

Fluoxetine hydrochloride（盐酸氟西汀）；olanzapine（奥氮平）170

Fluticasone furoate (糠酸氟替卡松酯)171

Fluticasone propionate（丙酸氟替卡松）171

Fluticasone propionate（丙酸氟替卡松）;salmeterol xinafoate（昔萘酸沙美特罗）174

Fluvastatin sodium（氟伐他汀钠）177

Fluvoxamine maleate (马来酸氟伏沙明)178

Follitropin alfa/beta (促卵泡生成素)178

Fomepizole (甲吡唑)180

Fomivirsen sodium（福米韦生钠）180

Formoterol fumarate (富马酸福莫特罗)180

Formoterol fumarate (富马酸福莫特罗);mometasone furoate(糠酸莫米松)181

Fosamprenavir calcium（福沙那韦钙）181

Fosaprepitant dimeglumine (福沙吡坦二甲葡胺)182

Fospropofol disodium (磷丙泊福钠)182

Frovatriptan succinate（琥珀酸夫罗曲坦）183

Fulvestrant（氟维司群）183

Gabapentin (加巴喷丁)184

Gabapentin enacarbil (加巴喷丁酯)185

Gadobutrol（钆布醇）185

Gadodiamide（钆双胺）185

Gadofosveset trisodium（钆磷维塞三钠）186

Gadoteridol（钆特醇）186

Gadoxetate disodium（钆塞酸二钠）187

Galantamine hydrobromide（氢溴酸加兰他敏）187

Gatifloxacin (加替沙星)187

Gefitinib（吉非替尼）188

Gemcitabine hydrochloride（吉西他滨）188

Gemifloxacin mesylate (甲磺酸吉米沙星)189

Gemtuzumab ozogamicin（吉妥单抗）189

Glatiramer acetate（醋酸格拉替雷）190

Glimepiride（格列美脲）; pioglitazone hydrochloride (盐酸吡格列酮)190

Glimepiride（格列美脲）;rosiglitazone maleate（马来酸罗格列酮）191

Glipizide（格列吡嗪）192

Glyburide （格列本脲）; metformin hydrochloride (盐酸二甲双胍)192

Glycopyrrolate (格隆溴铵)192

Goserelin acetate (醋酸戈舍瑞林)193

Granisetron hydrochloride（盐酸格拉司琼）193

Grepafloxacin hydrochloride（盐酸格帕沙星）194

Guaifenesin (愈创甘油醚)194

Guaifenesin（愈创甘油醚）; pseudoephedrine hydrochloride（盐酸伪麻黄碱）195

Guanfacine hydrochloride (盐酸胍法辛)195

Hexaminolevulinate hydrochloride (盐酸黑克斯胺)196

Histrelin acetate (醋酸组氨瑞林)196

Hyaluronidase recombinant human (重组人透明质酸酶)196

Hydralazine hydrochloride(盐酸肼屈嗪); isosorbide dinitrate（硝酸异山梨酯）197

Hydrochlorothiazide（氢氯噻嗪）; irbesartan（厄贝沙坦）197

Hydrochlorothiazide（氢氯噻嗪）; olmesartan medoxomil（奥美沙坦酯）198

Hydrochlorothiazide（氢氯噻嗪）; telmisartan（替米沙坦）198

Hydrochlorothiazide（氢氯噻嗪）; valsartan（缬沙坦）199

Hydrocodone bitartrate（酒石酸氢可酮）; ibuprofen（布洛芬）199

Hydromorphone hydrochloride (盐酸氢吗啡酮)199

Hydromorphone hydrochloride（盐酸氢吗啡酮）200

Hydroxocobalamin（羟钴胺）201

Ibandronate sodium (伊班膦酸钠)201

Ibuprofen (布洛芬)202

Ibuprofen lysine (布洛芬赖氨酸盐)202

Ibuprofen（布洛芬）; pseudoephedrine hydrochloride (盐酸伪黄麻碱)202

Icatibant acetate（醋酸艾替班特）203

Icodextrin（艾考糊精）203

Icosapent ethyl（二十碳五烯酸乙酯）203

Iloperidone（伊潘立酮）204

Imatinib mesylate（甲磺酸伊马替尼）204

Imiquimod(咪喹莫特)205

Indacaterol maleate (马来酸茚达特罗)205

Indinavir sulfate（硫酸茚地那韦）206

Indium In111 pentetreotide kit［铟（In111）喷曲肽］206

Ingenol mebutate (巨大戟醇甲基丁烯酸酯)207

Insulin aspart protamine recombinant （重组门冬胰岛素鱼精蛋白）; insulin aspart recombinant（重组门

冬胰岛素）207

Insulin aspart recombinant（重组门冬胰岛素）209

Insulin detemir recombinant（重组地特胰岛素）209

Insulin glargine recombinant (重组甘精胰岛素)210

Insulin glulisine recombinant (重组赖谷胰岛素)211

Insulin lispro protamine recombinant（重组赖脯胰岛素鱼精蛋白）; insulin lispro recombinant（重组赖脯胰岛素）212

Insulin lispro recombinant（重组赖脯胰岛素）213

Insulin recombinant human（重组人胰岛素）213

Ipratropium bromide（异丙托溴铵）214

Irbesartan（厄贝沙坦）214

Irinotecan hydrochloride（盐酸伊立替康）214

Iron dextran（右旋糖酐铁）215

Isotretinoin（异维A酸）215

Itraconazole（伊曲康唑）215

Ivacaftor (依瓦卡托)216

Ivermectin (伊维菌素)216

Ixabepilone (伊沙匹隆)217

Ketoconazole（酮康唑）218

Ketorolac tromethamine (酮洛酸氨丁三醇)218

Lacosamide（拉科酰胺）219

Lamivudine（拉米夫定）219

Lamivudine（拉米夫定）;zidovudine（齐多夫定）220

Lamotrigine (拉莫三嗪)220

Lanreotide acetate (醋酸兰瑞肽)220

Lansoprazole (兰索拉唑)221

Lanthanum carbonate（碳酸镧）221

Lapatinib ditosylate (对甲苯磺酸拉帕替尼)222

Lenalidomide (来那度胺)222

Leuprolide acetate（醋酸亮丙瑞林）224

Levalbuterol hydrochloride（盐酸左旋沙丁胺醇）226

Levalbuterol tartrate（酒石酸左旋沙丁胺醇）227

Levetiracetam (左乙拉西坦)227

Levobetaxololhydrochloride（盐酸倍他洛尔）227

Levobupivacaine hydrochloride（盐酸左布比卡因）228

Levocarnitine (左卡尼汀)228

Levocetirizine dihydrochloride（盐酸左西替利嗪）228

Levofloxacin (左氧氟沙星)229

Levoleucovorin calcium (左亚叶酸钙)229

Levonorgestrel（左炔诺孕酮）230

Levothyroxine sodium (左甲状腺素钠)230

Lidocaine（利多卡因）231

Lidocaine hydrochloride（盐酸利多卡因）232

Lidocaine（利卡多因）;prilocaine（丙胺卡因）232

Lidocaine（利卡多因）; tetracaine（丁卡因）232

Linaclotide（利那洛肽）233

Linagliptin (利拉利汀)233

Linagliptin（利拉利汀）; metformin hydrochloride(盐酸二甲双胍)234

Linezolid（利奈唑胺）235

Liraglutide recombinant (重组利拉鲁肽)235

Lisdexamfetamine dimesylate(二甲磺酸赖右苯丙胺)236

Lomitapide mesylate（甲磺酸洛美他派）238

Loperamide hydrochloride（盐酸洛哌丁胺）239

Loperamide hydrochloride（盐酸洛哌丁胺）; simethicone（二甲基硅油）239

Lopinavir（洛匹那韦）; ritonavir（利托那韦）240

Loratadine（氯雷他定）242

Loratadine（氯雷他定）;pseudoephedrine sulfate（硫酸伪麻黄碱）242

Lorcaserin hydrochloride（盐酸绿卡色林）243

Loteprednol etabonate（依碳酸氯替泼诺）243

Loteprednol etabonate（依碳酸氯替泼诺）; tobramycin（妥布霉素）244

Lovastatin（洛伐他汀）244

Lovastatin（洛伐他汀）;niacin（烟酸）245

Lubiprostone (鲁比前列酮)247

Lutropin alfa（促黄体素阿尔法）248

Magnesium chloride（氯化镁）; sodium bicarbonate（碳酸钠）;sodium chloride(氯化钠)248

Magnesium hydroxide（氢氧化镁）; omeprazole（奥美拉唑）; sodium bicarbonate（碳酸氢钠）249

Magnesium sulfate anhydrous （无水硫酸镁）; potassium sulfate（硫酸钾）; sodium sulfate (硫酸钠)249

Malathion (马拉硫磷)250

Mannitol（甘露醇）250

Maraviroc(马拉韦罗)250

Mecasermin recombinant（重组美卡舍明）251

Mecasermin rinfabate recombinant（重组美卡舍明里尼伐贝）251

Medroxyprogesterone acetate(醋酸甲羟孕酮)252

Megestrol acetate（醋酸甲地孕酮）252

Meloxicam (美洛昔康)252

Memantine hydrochloride (盐酸美金刚)252

Mequinol（甲氧苯酚）;tretinoin（维甲酸）253

Mesalamine (美沙拉嗪)253

Metaxalone (美他沙酮)254

Metformin hydrochloride（盐酸二甲双胍）254

Metformin hydrochloride（盐酸二甲双胍）; pioglitazone hydrochloride (盐酸吡格列酮)255

Metformin hydrochloride （盐酸二甲双胍）; repaglinide (瑞格列奈)256

Metformin hydrochloride（盐酸二甲双胍）;rosiglitazone maleate（马来酸罗格列酮）256

Metformin hydrochloride(盐酸二甲双胍); saxagliptin (沙格列汀)257

Metformin hydrochloride（盐酸双甲双胍）; sitagliptin phosphate (磷酸西他列汀)258

Methyl aminolevulinate hydrochloride（5氨基酮戊酸甲酯盐酸盐）259

Methylnaltrexone bromide（溴化甲基纳曲酮）259

Methylphenidate hydrochloride(盐酸哌甲酯)260

Metoclopramide hydrochloride（盐酸甲氧氯普胺）261

Metronidazole (甲硝唑)262

Micafungin sodium（米卡芬净钠）262

Miconazole(咪康唑)263

Miconazole nitrate（硝酸咪康唑）263

Milnacipran hydrochloride(盐酸米那普伦)263

Minocycline hydrochloride(盐酸米诺环素)264

Minoxidil (米诺地尔)265

Mirabegron（米拉贝龙）265

Mitomycin（丝裂霉素）266

Modafinil (莫达非尼)266

Mometasone furoate（糠酸莫米松）267

Mometasone furoate monohydrate（糠酸莫米松水合物）268

Montelukast sodium (孟鲁司特钠)268

Morphine sulfate(硫酸吗啡)269

Morphine sulfate(硫酸吗啡);naltrexone hydrochloride(盐酸纳曲酮)270

Moxifloxacin hydrochloride（盐酸莫西沙星）270

Mupirocin(莫匹罗星)271

Mupirocin calcium（莫匹罗星钙）271

Mycophenolate mofetil hydrochloride（盐酸吗替麦考酚酯）272

Mycophenolic acid（麦考酚酸）272

Naltrexone（纳曲酮）272

Naproxen sodium（萘普生钠）273

Naproxen sodium(萘普生钠);sumatriptan succinate(琥珀酸舒马普坦)273

Nateglinide（那格列奈）274

Nebivolol hydrochloride(盐酸奈必洛尔)274

Nelarabine（奈拉滨）275

Nelfinavir mesylate（甲磺奈非那韦）275

Nepafenac(奈帕芬胺)276

Nesiritide recombinant（重组奈西立肽）276

Niacin（烟酸）276

Niacin(烟酸);simvastatin(辛伐他汀)279

Nicardipine hydrochloride(盐酸尼卡地平)281

Nicotine（尼古丁）282

Nicotine polacrilex（尼古丁树脂）283

Nilotinib hydrochloride monohydrate(盐酸尼洛替尼水合物)283

Nisoldipine（尼索地平）284

Nizatidine(尼扎替丁)284

Nitric oxide（一氧化氮）284

Nitroglycerin（硝酸甘油）285

Nizatidine（尼扎替丁）286

Octreotide acetate（醋酸奥曲肽）286

Olanzapine(奥氮平)287

Olanzapine pamoate（奥氮平双羟萘酸）288

Olmesartan medoxomil（奥美沙坦酯）288

Olopatadine hydrochloride（盐酸奥洛他定）288

Omacetaxine mepesuccinate（高三尖杉酯碱）289

Omega3acid ethyl esters（omega3脂肪酸乙酯）289

Omeprazole（奥美拉唑）290

Omeprazole magnesium（奥美拉唑镁）290

Omeprazole（奥美拉唑）;sodium bicarbonate（碳酸氢钠）291

Ondansetron（昂丹司）292

Orlistat（奥利司他）292

Oseltamivir phosphate（磷酸奥司他韦）293

Oxaliplatin（奥沙利铂）293

Oxandrolone（氧雄龙）294

Oxcarbazepine（奥卡西平）295

Oxybutynin（奥昔布宁）295

Oxybutynin chloride（奥昔布宁氯）296

Oxycodone hydrochloride(盐酸羟考酮)297

Oxymorphone hydrochloride(盐酸羟吗啡酮)299

Paclitaxel(紫杉醇)301

Paliperidone palmitate(棕榈酸帕利哌酮)302

Palonosetron hydrochloride(盐酸帕洛诺司琼)303

Pancrelipase(胰脂肪酶)304

Pantoprazole sodium(泮托拉唑钠)304

Paricalcitol（帕立骨化醇）305

Paroxetine hydrochloride（盐酸帕罗西汀）306

Paroxetine mesylate（甲磺酸帕罗西汀）309

Pasireotide diaspartate（帕西瑞肽）310

Pazopanib hydrochloride(盐酸帕唑帕尼)310

Pegaptanib sodium（哌加他尼钠）311

Peginesatide acetate（聚乙二醇肽）311

Pegvisomant（培维索孟）312

Pemetrexed disodium(培美曲塞二钠)313

Penciclovir sodium（喷昔洛韦）313

Perampanel（吡仑帕奈）314

Perfluoropolymethylisopropyl ether（全氟聚甲基异丙基醚）;polytetrafluoroethylene（聚四氟乙烯）314

Perflutren（全氟丙烷）315

Phentermine hydrochloride(盐酸芬特明)315

Phentermine hydrochloride(盐酸芬特明);topiramate（托吡酯）315

Phentolamine mesylate（甲磺酸酚妥拉明）316

Pimecrolimus（吡美莫司）316

Pioglitazone hydrochloride（盐酸吡格列酮）317

Piperacillin sodium(哌拉西林钠);tazobactam sodium(他唑巴坦钠)317

Pitavastatin calcium(匹伐他汀钙)318

Plerixafor(普乐沙福)319

Ponatinib hydrochloride（盐酸普纳替尼）319

Posaconazole（泊沙康唑）320

Pralatrexate(普拉曲沙)320

Pramipexole dihydrochloride(盐酸普拉克索)320

Pramlintide acetate（醋酸普兰林肽）321

Prasugrel hydrochloride(盐酸普拉格雷)322

Pravastatin sodium（普伐他汀钠）322

Prednisolone acetate(醋酸泼尼松龙)323

Prednisolone sodium phosphate(泼尼松龙磷酸钠)323

Prednisone（泼尼松）324

Pregabalin（普瑞巴林）324

Progesterone(黄体酮)325

Propafenone hydrochloride（盐酸普罗帕酮）326

Propofol（丙泊酚）326

Propranolol hydrochloride(盐酸普萘洛尔)327

Quazepam(夸西泮)327

Quetiapine fumarate（富马酸喹硫平）327

Quinapril hydrochloride（盐酸喹那普利）328

Rabeprazole sodium（雷贝拉唑钠）328

Raloxifene hydrochloride（盐酸雷洛昔芬）329

Raltegravir potassium(雷特格韦钾)329

Ramelteon（拉米替隆）330

Ramipril(雷米普利)330

Ranitidine bismuth citrate（枸橼酸铋雷尼替丁）331

Ranolazine（雷诺嗪）331

Rasagiline mesylate(甲磺酸雷沙吉兰)331

Regadenoson(瑞加德松)332

Regorafenib（瑞格菲尼）332

Remifentanil hydrochloride(盐酸瑞芬太尼)333

Repaglinide（瑞格列奈）333

Retapamulin(瑞他莫林)333

Ribavirin（利巴韦林）334

Rifaximin(利福昔明)335

Rilpivirine hydrochloride(盐酸瑞丽匹维)336

Risedronate sodium(利塞膦酸钠)336

Risperidone(利培酮)337

Ritonavir(利托那韦)340

Rivaroxaban(利伐沙班)341

Rivastigmine(利伐斯的明)342

Rizatriptan benzoate(苯甲酸利扎曲普坦)343

Rofecoxib(罗非昔布)343

Roflumilast(罗氟司特)345

Romidepsin(罗米内酯)345

Ropinirole hydrochloride(盐酸罗匹尼罗)345

Ropivacaine hydrochloride(盐酸罗哌卡因)346

Rosiglitazone maleate(马来酸罗格列酮)346

Rosuvastatin calcium(瑞舒伐他汀钙)347

Rotigotine(罗替戈汀)348

Rufinamide(卢非酰胺)349

Ruxolitinib phosphate(膦酸罗克斯替尼)350

Salmeterol xinafoate(昔萘酸沙美特罗)350

Sapropterin dihydrochloride(盐酸沙丙蝶呤)350

Saquinavir mesylate(甲磺酸沙奎那韦)351

Saxagliptin hydrochloride(盐酸沙格列汀)351

Selegiline(司来吉兰)351

Sertaconazole nitrate(硝酸舍他康唑)352

Sertraline hydrochloride(盐酸舍曲林)352

Sevelamer carbonate(碳酸司维拉姆)353

Sevelamer hydrochloride(盐酸司维拉姆)353

Sevoflurane(七氟烷)354

Sibutramine hydrochloride(盐酸西布曲明)354

Sildenafil citrate(枸橼酸西地那非)355

Silodosin(西罗多辛)355

Simvastatin(辛伐他汀)；sitagliptin phosphate(磷酸西格列汀)355

Sincalide(辛卡利特)357

Sinecatechins(西勒茶素)358

Sirolimus(西罗莫司)358

Sitagliptin phosphate(磷酸西他列汀)359

Sodium oxybate(羟丁酸钠)361

Sodium phosphate, dibasic anhydrous(无水磷酸二钠);sodium phosphate monobasic monohydrate

(磷酸二氢钠单水合物)361

Solifenacin succinate(琥珀酸索非那新)362

Somatropin recombinant（重组人生长激素）362

Sorafenib tosylate(甲苯磺酸索拉非尼)365

Spinosad(多杀菌素)365

Stavudine（司他夫定）365

Sumatriptan（舒马曲坦）366

Sumatriptan succinate（舒马坦琥珀酸盐）366

Sunitinib malate(苹果酸舒尼替尼)367

Tacrolimus（他克莫司）367

Tadalafil（他达拉非）368

Taliglucerase alfa（它利罗酶）368

Tamoxifen citrate（枸橼酸他莫昔芬）369

Tapentadol hydrochloride（盐酸他喷他多）369

Tazarotene（他扎罗汀）371

Technetium Tc99m apcitide（阿匹西肽锝99m）371

Technetium Tc99m mertiatide kit（巯替肽锝99m）371

Technetium Tc99m Teboroxime Kit(替肟锝试剂盒)371

Teduglutide recombinant（替度鲁肽）372

Tegaserod maleate（马来酸替加色罗）372

Telaprevir(特拉匹韦)372

Telavancin hydrochloride(盐酸特拉万星)373

Telbivudine(替比夫定)373

Telithromycin（泰利霉素）374

Telmisartan(替米沙坦)374

Temozolomide(替莫唑胺)375

Temsirolimus(坦罗莫司)375

Tenofovir disoproxil fumarate（替诺福韦酯富马酸盐）376

Terazosin hydrochloride（盐酸特拉唑嗪）378

Terbinafine（特比萘芬）378

Teriflunomide（特立氟胺）379

Teriparatide recombinant human（人重组特立帕肽）379

Tesamorelin acetate(醋酸替莫瑞林)380

Testosterone(睾丸素)380

Thalidomide（沙利度胺）381

Thyrotropin alfa（促甲状腺素α）383

Tiagabine hydrochloride（盐酸噻加宾）384

Ticagrelor(替卡格雷)384

Tigecycline(替加环素)384

Timolol maleate(马来酸噻吗洛尔)385

Tiotropium bromide monohydrate(噻托溴铵一水合物)385

Tipranavir(替拉那韦)386

Tirofiban hydrochloride（盐酸替罗非班）386

Tobramycin（妥布霉素）387

Tofacitinib citrate（枸橼酸托法替尼）387

Tolterodine tartrate（酒石酸托特罗定）388

Tolvaptan（托伐普坦）388

Topiramate（托吡酯）389

Topotecan hydrochloride（盐酸拓扑替康）390

Tramadol hydrochloride(盐酸曲马多)391

Trandolapril（群多普利）391

Trandolapril（群多普利）; verapamil hydrochloride（盐酸维拉帕米）392

Tranexamic acid(氨甲环酸)392

Travoprost（曲伏前列素）392

Trazodone hydrochloride(盐酸曲唑酮)393

Treprostinil sodium(曲前列尼尔钠)393

Tretinoin(维A酸)394

Triamcinolone acetonide（曲安奈德）394

Trimethoprim hydrochloride（盐酸甲氧苄啶）395

Trimetrexate glucuronate（葡萄糖醛酸三甲曲沙）395

Triptorelin pamoate（羟萘酸曲普瑞林）395

Troglitazone（曲格列酮）396

Trospium chloride(曲司氯铵)396

Trovafloxacin mesylate（甲磺酸曲伐沙星）397

Unoprostone isopropyl(乌诺前列酮异丙酯)397

Urofollitropin（尿促卵泡素）398

Valacyclovir hydrochloride（盐酸伐昔洛韦）398

Valdecoxib（伐地昔布）398

Valganciclovir hydrochloride（缬更昔洛韦盐酸盐）399

Valsartan（缬沙坦）399

Vandetanib(凡德他尼)400

Vardenafil hydrochloride（盐酸伐地那非）400

Varenicline tartrate（酒石酸伐尼克兰）401

Vemurafenib(威罗菲尼)401

Venlafaxine hydrochloride（盐酸文法拉辛）402

Verapamil hydrochloride（盐酸维拉帕米）403

Verteporfin（维替泊芬）403

Vilazodone hydrochloride(盐酸维拉佐酮)404

Vincristine sulfate（硫酸长春新碱）404

Vismodegib（维莫德吉）405

Voriconazole（伏立康唑）405

Vorinostat(伏立诺他)405

Zafirlukast（扎鲁司特）406

Zanamivir（扎那米韦）406

Ziconotide（齐可诺肽）407

Zileuton（齐留通）407

Ziprasidone hydrochloride（盐酸齐拉西酮）407

Zoledronic acid(唑来磷酸)408

Zolmitriptan（佐米曲普坦）408

Zolpidem tartrate(酒石酸唑吡坦)409

附录1：专利药品常见剂型中英文对照表410

附录2：美国药品市场独占权代码定义414

附录3：美国药品市场独占权代码定义454

中文索引482

本书主要介绍了截至2013年5月，美国批准上市的药品中所有受专利和行政保护（即市场独占权保护）的药品。全书按药物活性成分的英文字母顺序进行编排。针对每一个药品,本书设立了药品名称、药品简介、药品的专利和行政保护情况版块。全书大量采用表格，简明扼要，力求以最小的篇幅囊括最大量的药品信息，方便读者查阅。本书所收集的专利可在一定程度上反映出全球最新、最前沿和实用的医药科技发展水平。全书共涉及药物活性成分700余种,各种药品制剂共4000多种，药品专利10000多项。
本书的读者对象为:任何打算合法仿制美国药品和希望了解美国上市药品的专利保护情况的企业和个人；任何有意从现有的最新、最前沿和实用的药品专利技术中寻找灵感和启发的医药科学人员；制药企业的科研人员和管理人员；各级政府与药品有关的管理决策人员,关心国外医药信息的情报人员；大专院校、科研机构中所有与药品研究开发有关的大学高年级本科生、研究生、 科技工作者等。

作者长期工作在新药研究的第一线，紧密跟踪国外医药科研的最前沿，了解医药科研领域类的最先进的技术、成果和发展动向。《美国药品专利与行政保护速查》主要介绍了截止2013年5月为止，受到专利和行政保护的美国药品，资料新、内容全，以表格形式呈现，方便查阅。